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3 Contraception

Contraceptives, hormonal

Overview

The Fraser Guidelines (Department of Health Guidance (July

2004): Best practice guidance for doctors and other health

professionals on the provision of advice and treatment to

young people under 16 on contraception, sexual and

reproductive health, available at www.tinyurl.com/bpg16)

should be followed when prescribing contraception for

women under 16 years. The UK Medical Eligibility Criteria for

Contraceptive Use (available at www.fsrh.org) is published by

the Faculty of Sexual and Reproductive Healthcare; it

categorises the risks of using contraceptive methods with

pre-existing medical conditions.

Hormonal contraception is the most effective method of

fertility control, but can have major and minor side-effects,

especially for certain groups of women. Hormonal

contraception should only be used by adolescents after

menarche.

Intra-uterine devices are a highly effective method of

contraception but may produce undesirable local sideeffects. They may be used in women of all ages irrespective

of parity, but are less appropriate for those with an increased

risk of pelvic inflammatory disease.

Barrier methods alone (condoms, diaphragms, and caps)

are less effective but can be reliable for well-motivated

couples if used in conjunction with a spermicide.

Occasionally sensitivity reactions occur. A female condom

(Femidom®) is also available; it is pre-lubricated but does not

contain a spermicide.

Combined hormonal contraceptives

Oral contraceptives containing an oestrogen and a

progestogen (‘combined oral contraceptives’) are effective

preparations for general use. Advantages of combined oral

contraceptives include:

. reliable and reversible;

. reduced dysmenorrhoea and menorrhagia;

. reduced incidence of premenstrual tension;

. less symptomatic fibroids and functional ovarian cysts;

. less benign breast disease;

. reduced risk of ovarian and endometrial cancer;

. reduced risk of pelvic inflammatory disease.

Combined oral contraceptives containing a fixed amount

of an oestrogen and a progestogen in each active tablet are

termed ‘monophasic’; those with varying amounts of the two

hormones are termed ‘phasic’. A transdermal patch and a

vaginal ring, both containing an oestrogen with a

progestogen, are also available.

Combined Oral Contraceptives Monophasic

21-day preparations

Oestrogen

content

Progestogen

content

Brand

Ethinylestradiol

20 micrograms

Desogestrel

150 micrograms

Gedarel® 20/150

Ethinylestradiol

20 micrograms

Desogestrel

150 micrograms

Mercilon®

Ethinylestradiol

20 micrograms

Gestodene

75 micrograms

Femodette®

Ethinylestradiol

20 micrograms

Gestodene

75 micrograms

Millinette® 20/75

Ethinylestradiol

20 micrograms

Gestodene

75 micrograms

Sunya® 20/75

Ethinylestradiol

20 micrograms

Norethisterone

acetate 1 mg

Loestrin® 20

Ethinylestradiol

30 micrograms

Desogestrel

150 micrograms

Gedarel® 30/150

Ethinylestradiol

30 micrograms

Desogestrel

150 micrograms

Marvelon®

Ethinylestradiol

30 micrograms

Drospirenone 3 mg Yasmin®

Ethinylestradiol

30 micrograms

Gestodene

75 micrograms

Femodene®

Ethinylestradiol

30 micrograms

Gestodene

75 micrograms

Katya® 30/75

Ethinylestradiol

30 micrograms

Gestodene

75 micrograms

Millinette® 30/75

Ethinylestradiol

30 micrograms

Levonorgestrel

150 micrograms

Levest®

Ethinylestradiol

30 micrograms

Levonorgestrel

150 micrograms

Microgynon® 30

Ethinylestradiol

30 micrograms

Levonorgestrel

150 micrograms

Ovranette®

Ethinylestradiol

30 micrograms

Levonorgestrel

150 micrograms

Rigevidon®

Ethinylestradiol

30 micrograms

Norethisterone

acetate 1.5 mg

Loestrin® 30

Ethinylestradiol

35 micrograms

Norgestimate

250 micrograms

Cilest®

Ethinylestradiol

35 micrograms

Norethisterone

500 micrograms

Brevinor®

Ethinylestradiol

35 micrograms

Norethisterone 1 mg Norimin®

Mestranol

50 micrograms

Norethisterone 1 mg Norinyl-1®

Combined Oral Contraceptives Monophasic

28-day preparations

Oestrogen

content

Progestogen

content

Brand

Ethinylestradiol

30 micrograms

Gestodene

75 micrograms

Femodene® ED

Ethinylestradiol

30 micrograms

Levonorgestrel

150 micrograms

Microgynon® 30 ED

Estradiol (as

hemihydrate)

1.5 mg

Nomegestrol acetate

2.5 mg

Zoely®

BNF 78 Contraception 791

Genito-urinary system

7

Combined Oral Contraceptives Phasic 21-day

preparations

Oestrogen content Progestogen content Brand

Ethinylestradiol

30 micrograms

Levonorgestrel

50 micrograms

Logynon Ethinylestradiol ®

40 micrograms

Levonorgestrel

75 micrograms

Ethinylestradiol

30 micrograms

Levonorgestrel

125 micrograms

Ethinylestradiol

30 micrograms

Levonorgestrel

50 micrograms

TriRegol Ethinylestradiol ®

40 micrograms

Levonorgestrel

75 micrograms

Ethinylestradiol

30 micrograms

Levonorgestrel

125 micrograms

Ethinylestradiol

35 micrograms

Norethisterone

500 micrograms

Synphase Ethinylestradiol ®

35 micrograms

Norethisterone 1 mg

Ethinylestradiol

35 micrograms

Norethisterone

500 micrograms

Combined Oral Contraceptives Phasic 28-day

preparations

Oestrogen

content

Progestogen

content

Brand

Ethinylestradiol

30 micrograms

Levonorgestrel

50 micrograms

Logynon® ED Ethinylestradiol

40 micrograms

Levonorgestrel

75 micrograms

Ethinylestradiol

30 micrograms

Levonorgestrel

125 micrograms

Estradiol valerate

3 mg

Qlaira®

Estradiol valerate

2 mg

Dienogest 2 mg

Estradiol valerate

2 mg

Dienogest 3 mg

Estradiol valerate

1 mg

Choice

The majority of combined oral contraceptives contain

ethinylestradiol p. 759 as the oestrogen component;

mestranol and estradiol are also used. The ethinylestradiol

content of combined oral contraceptives ranges from 20 to

40 micrograms. Generally a preparation with the lowest

oestrogen and progestogen content which gives good cycle

control and minimal side-effects in the individual woman is

chosen. It is recommended that combined hormonal

contraceptives are not continued beyond 50 years of age

since more suitable alternatives exist.

. Low strength preparations (containing ethinylestradiol

20 micrograms) are particularly appropriate for women

with risk factors for circulatory disease, provided a

combined oral contraceptive is otherwise suitable.

. Standard strength preparations (containing ethinylestradiol

30 or 35 micrograms or in 30–40 microgram phased

preparations) are appropriate for standard use. Phased

preparations are generally reserved for women who either

do not have withdrawal bleeding or who have

breakthrough bleeding with monophasic products.

The progestogens ethinylestradiol with desogestrel p. 798,

ethinylestradiol with drospirenone p. 798, and

ethinylestradiol with gestodene p. 799 may be considered for

women who have side-effects (such as acne, headache,

depression, breast symptoms, and breakthrough bleeding)

with other progestogens. Drospirenone, a derivative of

spironolactone, has anti-androgenic and antimineralocorticoid activity; it should be used with care if an

increased plasma-potassium concentration might be

hazardous.

Dienogest with estradiol valerate p. 797 is in the combined

oral contraceptive Qlaira ®. Nomegestrol is the progestogen

contained in the combined oral contraceptive Zoely ®, in

combination with estradiol.

The progestogen norelgestromin is combined with

ethinylestradiol in a transdermal patch (Evra ®). The vaginal

contraceptive ring contains the progestogen etonogestrel

combined with ethinylestradiol (NuvaRing ®).

Surgery

Oestrogen-containing contraceptives should preferably be

discontinued (and adequate alternative contraceptive

arrangements made) 4 weeks before major elective surgery

and all surgery to the legs or surgery which involves

prolonged immobilisation of a lower limb; they should

normally be recommenced at the first menses occurring at

least 2 weeks after full mobilisation. A progestogen-only

contraceptive may be offered as an alternative and the

oestrogen-containing contraceptive restarted after

mobilisation. When discontinuation of an oestrogencontaining contraceptive is not possible, e.g. after trauma or

if a patient admitted for an elective procedure is still on an

oestrogen- containing contraceptive, thromboprophylaxis

(with unfractionated or low molecular weight heparin and

graduated compression hosiery) is advised. These

recommendations do not apply to minor surgery with short

duration of anaesthesia, e.g. laparoscopic sterilisation or

tooth extraction, or to women using oestrogen-free

hormonal contraceptives.

Reason to stop immediately

Combined hormonal contraceptives or hormone

replacement therapy (HRT) should be stopped (pending

investigation and treatment), if any of the following occur:

. sudden severe chest pain (even if not radiating to left

arm);

. sudden breathlessness (or cough with blood-stained

sputum);

. unexplained swelling or severe pain in calf of one leg;

. severe stomach pain;

. serious neurological effects including unusual severe,

prolonged headache especially if first time or getting

progressively worse or sudden partial or complete loss of

vision or sudden disturbance of hearing or other

perceptual disorders or dysphasia or bad fainting attack or

collapse or first unexplained epileptic seizure or weakness,

motor disturbances, very marked numbness suddenly

affecting one side or one part of body;

. hepatitis, jaundice, liver enlargement;

. blood pressure above systolic 160 mmHg or diastolic

95 mmHg; (in adolescents stop if blood pressure very

high);

. prolonged immobility after surgery or leg injury;

. detection of a risk factor which contra-indicates

treatment.

Progestogen-only contraceptives

Oral progestogen-only contraceptives

Oral progestogen-only preparations alter cervical mucus to

prevent sperm penetration and may inhibit ovulation in

some women; oral desogestrel-only preparations

consistently inhibit ovulation and this is their primary

mechanism of action. There is insufficient clinical trial

evidence to compare the efficacy of oral progestogen-only

contraceptives with each other or with combined hormonal

792 Contraception BNF 78

Genito-urinary system

7

contraceptives. Progestogen-only contraceptives offer a

suitable alternative to combined hormonal contraceptives

when oestrogens are contra-indicated (including those with

venous thrombosis or a past history or predisposition to

venous thrombosis, heavy smokers, those with hypertension

above systolic 160 mmHg or diastolic 95 mmHg, valvular

heart disease, diabetes mellitus with complications, and

migraine with aura).

Parenteral progestogen-only contraceptives

Medroxyprogesterone acetate p. 810 (Depo-Provera ®,

SAYANA PRESS ®) is a long-acting progestogen given by

injection; it is at least as effective as the combined oral

preparations but because of its prolonged action it should

never be given without full counselling backed by the patient

information leaflet. It may be used as a short-term or longterm contraceptive for women who have been counselled

about the likelihood of menstrual disturbance and the

potential for a delay in return to full fertility. Delayed return

of fertility and irregular cycles may occur after

discontinuation of treatment but there is no evidence of

permanent infertility. Troublesome bleeding has been

reported in patients given medroxyprogesterone acetate in

the immediate puerperium; delaying the first injection until

6 weeks after birth may minimise bleeding problems. If the

woman is not breast-feeding, the first injection may be given

within 5 days postpartum (she should be warned that the risk

of troublesome bleeding may be increased).

. In adolescents, medroxyprogesterone acetate (DepoProvera ®, SAYANA PRESS ®) should be used only when

other methods of contraception are inappropriate;

. in all women, the benefits of using medroxyprogesterone

acetate beyond 2 years should be evaluated against the

risks;

. in women with risk factors for osteoporosis, a method of

contraception other than medroxyprogesterone acetate

should be considered.

Norethisterone enantate (Noristerat ®) is a long-acting

progestogen given as an oily injection which provides

contraception for 8 weeks; it is used as short-term interim

contraception e.g. before vasectomy becomes effective.

An etonogestrel-releasing implant (Nexplanon ®) is also

available. It is a highly effective long-acting contraceptive,

consisting of a single flexible rod that is inserted

subdermally into the lower surface of the upper arm and

provides contraception for up to 3 years. The manufacturer

advises that in heavier women, blood-etonogestrel

concentrations are lower and therefore the implant may not

provide effective contraception during the third year; they

advise that earlier replacement may be considered in such

patients—however, evidence to support this

recommendation is lacking. Local reactions such as bruising

and itching can occur at the insertion site. The contraceptive

effect of etonogestrel is rapidly reversed on removal of the

implant.

Intra-uterine progestogen-only device

The progestogen-only intra-uterine systems Mirena ®,

Jaydess ® and Levosert ® release levonorgestrel p. 806 directly

into the uterine cavity. Mirena ® is licensed for use as a

contraceptive, for the treatment of primary menorrhagia and

for the prevention of endometrial hyperplasia during

oestrogen replacement therapy. Jaydess ® and Levosert ® are

licensed for contraception, and Levosert ® is additionally

licensed for the treatment of menorrhagia. These may

therefore be a contraceptive method of choice for women

who have excessively heavy menses.

The effects of the progestogen-only intra-uterine system

are mainly local and hormonal including prevention of

endometrial proliferation, thickening of cervical mucus, and

suppression of ovulation in some women (in some cycles). In

addition to the progestogenic activity, the intra-uterine

system itself may contribute slightly to the contraceptive

effect. Return of fertility after removal is rapid and appears

to be complete.

Advantages of the progestogen-only intra-uterine system

over copper intra-uterine devices are that there may be an

improvement in any dysmenorrhoea and a reduction in

blood loss; there is also evidence that the frequency of pelvic

inflammatory disease may be reduced (particularly in the

youngest age groups who are most at risk).

In primary menorrhagia, menstrual bleeding is reduced

significantly within 3–6 months of inserting the

progestogen-only intra-uterine system, probably because it

prevents endometrial proliferation. Another treatment

should be considered if menorrhagia does not improve

within this time.

Surgery

All progestogen-only contraceptives (including those given

by injection) are suitable for use as an alternative to

combined hormonal contraceptives before major elective

surgery, before all surgery to the legs, or before surgery

which involves prolonged immobilisation of a lower limb.

Contraceptives, non-hormonal

Spermicidal contraceptives

Spermicidal contraceptives are useful additional safeguards

but do not give adequate protection if used alone unless

fertility is already significantly diminished. They have two

components: a spermicide and a vehicle which itself may

have some inhibiting effect on sperm activity. They are

suitable for use with barrier methods, such as diaphragms or

caps; however, spermicidal contraceptives are not generally

recommended for use with condoms, as there is no evidence

of any additional protection compared with non-spermicidal

lubricants.

Spermicidal contraceptives are not suitable for use in

those with or at high risk of sexually transmitted infections

(including HIV); high frequency use of the spermicide

nonoxinol ‘9’ p. 811 has been associated with genital lesions,

which may increase the risk of acquiring these infections.

Contraceptive devices

Intra-uterine devices

The intra-uterine device (IUD) is a suitable contraceptive for

women of all ages irrespective of parity; however, it is less

appropriate for those with an increased risk of pelvic

inflammatory disease e.g. women under 25 years.

The most effective intra-uterine devices have at least

380 mm2 of copper and have banded copper on the arms.

Smaller devices have been introduced to minimise sideeffects; these consist of a plastic carrier wound with copper

wire or fitted with copper bands; some also have a central

core of silver to prevent fragmentation of the copper.

Fertility declines with age and therefore a copper intrauterine device which is fitted in a woman over the age of 40,

may remain in the uterus until menopause.

A frameless, copper-bearing intra-uterine device (Gyne

Fix ®) is also available. It consists of a knotted, polypropylene

thread with 6 copper sleeves; the device is anchored in the

uterus by inserting the knot into the uterine fundus.

Caution with oil-based lubricants

Products such as petroleum jelly (Vaseline ®), baby oil and

oil-based vaginal and rectal preparations are likely to

damage condoms and contraceptive diaphragms made from

latex rubber, and may render them less effective as a barrier

method of contraception and as a protection from sexually

transmitted infections (including HIV).

BNF 78 Contraception 793

Genito-urinary system

7

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